SCHEMBL4581908

SCHEMBL4581908

O=C1NCCN(c2nc(Cl)ncc2Br)C1c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 14/20 0.42
BCR P11274 14/20 0.42
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
MAPT P10636 1/20 0.35
SCN9A Q15858 1/20 0.35
RPS6KA5 O75582 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4581852 0.79 IDH1 (0.44)
SCHEMBL4581848 0.79 IDH1 (0.44)
SCHEMBL4591653 0.79 HDAC1 (0.40) HDAC1HDAC8HDAC6SCN9ARPS6KA5
SCHEMBL10506257 0.71 RXFP1 (0.44)
SCHEMBL4580829 0.69 HDAC1 (0.42) HDAC1HDAC8HDAC6MAPT
SCHEMBL4581847 0.68 HDAC1 (0.43) HDAC1HDAC8HDAC6MAPT
SCHEMBL4581690 0.68 TRPV1 (0.42) HDAC1HDAC8HDAC6MAPT
SCHEMBL21361176 0.67 CDK4 (0.40) ABL1BCRMAPT
SCHEMBL4580841 0.67 IDH1 (0.42) HDAC1HDAC8HDAC6
SCHEMBL4580975 0.67 IKBKB (0.41) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US disclosed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080258-A1 Pyridine and pyrimidine derivatives ROR1, MAPK1, IRAK1 ABL1 32/4885BCR 63/4885HDAC1 481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.