SCHEMBL4582646

SCHEMBL4582646

COc1ccc(C[C@@H](N)CN2C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.60
KMT2A Q03164 2/20 0.56
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.52
RPS6KA2 Q15349 2/20 0.51
NR1H3 Q13133 1/20 0.51
GAA P10253 2/20 0.49
MEN1 O00255 1/20 0.49
APAF1 O14727 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4582642 1.00 CASP3 (0.60) CASP3KMT2ANPC1RAB9ARPS6KA2
SCHEMBL4784027 0.85 TAAR1 (0.55) CASP3KMT2ANPC1RAB9ANR1H3
SCHEMBL13919633 0.85 CASP3 (0.44) CASP3KMT2ANPC1RAB9ARPS6KA2
Hydrochloric Acid SCHEMBL4899590 0.84 TAAR1 (0.54) CASP3KMT2ANPC1NR1H3GAA
SCHEMBL1529483 0.84 EPHX1 (0.53) CASP3GAA
SCHEMBL2370243 0.84 EPHX1 (0.53) CASP3GAA
SCHEMBL1529481 0.84 EPHX1 (0.53) CASP3GAA
Hydrochloric Acid SCHEMBL1529614 0.82 EPHX1 (0.52) CASP3GAA
Hydrochloric Acid SCHEMBL4778820 0.82 EPHX1 (0.52) CASP3GAA
Hydrochloric Acid SCHEMBL4783273 0.82 EPHX1 (0.52) CASP3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed