SCHEMBL4582835

SCHEMBL4582835

Cc1ccccc1CNS

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.55
HPGD P15428 3/20 0.50
ALDH1A1 P00352 3/20 0.50
TAAR1 Q96RJ0 1/20 0.48
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
HTT P42858 2/20 0.46
GAA P10253 2/20 0.46
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.43
ACHE P22303 1/20 0.43
DNM1 Q05193 1/20 0.42
CYP2A13 Q16696 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL40401 0.82 CHRM2 (0.69) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL606716 0.80 CHRM2 (0.55) CHRM2HPGDALDH1A1TAAR1KMT2A
Hydrochloric Acid SCHEMBL6065696 0.80 CHRM2 (0.67) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL6896147 0.78 CHRM2 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL6784532 0.78 ALDH1A1 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A
Hydrochloric Acid SCHEMBL23527967 0.78 CHRM2 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL9995162 0.78 CHRM2 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL24170552 0.78 CHRM2 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL8014820 0.78 CHRM2 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A
SCHEMBL15129253 0.78 CHRM2 (0.53) CHRM2HPGDALDH1A1TAAR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022000443-A1 METHODS AND COMPOSITIONS FOR TARGETING TREGS USING CCR8 INHIBITORS Nanjing Immunophage Biotech Co., Ltd. (CN) 2022-01-06 WO disclosed
CN-107074866-B Pyrimido-pyrrole compound, preparation method thereof, medicinal composition and application thereof 厦门大学 2019-06-07 CN disclosed
EP-2632460-B1 THIOPHENE DERIVATIVES FOR USE IN THE TREATMENT OF TUBERCULOSIS UNIV VIRGINIA PATENT FOUNDATION (US) 2018-02-28 EP disclosed
CN-107074866-A Pyrimido-pyrrole compound, preparation method thereof, medicinal composition and application thereof 厦门大学 2017-08-18 CN disclosed
CN-106188060-A Pyrimido azoles, its preparation method, Pharmaceutical composition and application thereof 厦门大学 2016-12-07 CN disclosed
CN-101400336-B Novel flavoring agents, taste modifiers, tastants, taste enhancers, umami or sweeteners and/or enhancers and uses thereof SENOMYX INC 2013-06-05 CN disclosed
CN-101400336-A Novel flavoring agents, taste modifiers, tastants, taste enhancers, umami or sweeteners and/or enhancers and uses thereof SENOMYX INC (US) 2009-04-01 CN disclosed
CN-101203142-A Aromatic amides and ureas and their uses as sweet and/or delicate flavor modifiers, flavouring agents and taste enhancers SENOMYX INC (US) 2008-06-18 CN disclosed
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US disclosed
CN-1301981-C Medicinal composition containing 1,3-thiazine derivative SHIONOGI & CO (JP) 2007-02-28 CN disclosed
CN-1247553-C 2-imino-1,3-thiazine derivs. SHIONOGI & CO (JP) 2006-03-29 CN disclosed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US disclosed
EP-1448555-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES Celltech R & D Limited (GB) 2004-08-25 EP disclosed
WO-2003045941-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES CELLTECH R & D LIMITED (GB) 2003-06-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080258-A1 Pyridine and pyrimidine derivatives ROR1, MAPK1, IRAK1 CHRM2 861/4885HPGD 1994/4885ALDH1A1 682/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.