SCHEMBL458327

SCHEMBL458327

C=CC(N)O[PH](=O)OC(N)C=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL458328 0.79
SCHEMBL9303806 0.74
SCHEMBL788280 0.67
SCHEMBL1533439 0.67
SCHEMBL6403967 0.67
SCHEMBL11496566 0.67
SCHEMBL11636625 0.67
SCHEMBL170397 0.65
SCHEMBL10596901 0.65
SCHEMBL11496567 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 176 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9738895-B2 Oligomeric compounds and methods IONIS PHARMACEUTICALS, INC. (US) 2017-08-22 US claimed
CN-104031086-B Method for synthesizing alpha-amino alkyl phosphonate compounds 湖南大学 2017-05-10 CN claimed
US-20150167006-A1 OLIGOMERIC COMPOUNDS AND METHODS ISIS PHARMACEUTICALS, INC. (US) 2015-06-18 US claimed
US-8987435-B2 Oligomeric compounds and methods ISIS PHARMACEUTICALS, INC. (US) 2015-03-24 US claimed
CN-104031086-A Method for synthesizing alpha-amino alkyl phosphonate compounds UNIV HUNAN 2014-09-10 CN claimed
US-8512976-B2 Selective growth media OXOID LIMITED (GB) 2013-08-20 US claimed
EP-2447274-A2 Oligomeric compounds and methods Isis Pharmaceuticals, Inc. (US) 2012-05-02 EP claimed
US-20110313019-A1 OLIGOMERIC COMPOUNDS AND METHODS ISIS PHARMACEUTICALS, INC. (US) 2011-12-22 US claimed
EP-2358398-A2 OLIGOMERIC COMPOUNDS AND METHODS Isis Pharmaceuticals, Inc. (US) 2011-08-24 EP claimed
US-20100248331-A1 SELECTIVE GROWTH MEDIA DRUGGAN PATRICK 2010-09-30 US claimed
WO-2010048585-A2 OLIGOMERIC COMPOUNDS AND METHODS ISIS PHARMACEUTICALS, INC. (US) 2010-04-29 WO claimed
EP-1334175-B1 IMPROVEMENTS IN OR RELATING TO SELECTIVE AGENTS FOR BIOLOGICAL CULTURES OXOID LTD (GB) 2009-12-23 EP claimed
CN-1282653-C Fluoric alpha-aminoalkyl phosphonate with agricultural antiviral activity and its synthesis UNIV GUIZHOU (CN) 2006-11-01 CN claimed
CN-1432573-A Fluoric alpha-aminoalkyl phosphonate with agricultural antiviral activity and its synthesis UNIV GUIZHOU (CN) 2003-07-30 CN claimed
WO-1995031572-A1 AMINOHYDROCARBON PHOSPHONATE OLIGONUCLEOTIDES AND USES THEREFOR PHARMGENICS, INC. (US) 1995-11-23 WO claimed
US-20240229029-A9 COMPOSITIONS AND METHODS FOR TREATMENT OF FRIEDREICH'S ATAXIA THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-07-11 US disclosed
US-20240141348-A1 ALLELE SELECTIVE INHIBITION OF MUTANT C9ORF72 FOCI EXPRESSION BY DUPLEX RNAS TARGETING THE EXPANDED HEXANUCLEOTIDE REPEAT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-05-02 US disclosed
US-4795632-A ACRYLALDEHYDE-ACRYLIC ACID COPOLYMER AND PHOSPHATE OR PHOSPHONATE HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1989-01-03 US disclosed
EP-0253179-A2 A-acylamino aminoalkyl phophonate angiotensin converting enzyme inhibitors E.R. Squibb &amp; Sons, Inc. (US) 1988-01-20 EP disclosed
US-4013813-A AMINOALKYLPHOSPHONIC ACID ESTER-BASED TEXTILE FIRE RETARDANTS LEBLANC RESEARCH CORPORATION (US) 1977-03-22 US disclosed