SCHEMBL4583314

SCHEMBL4583314

CCCCCOc1ccn(CCCCNS(C)(=O)=O)c(=O)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MCHR1 Q99705 6/20 0.40
KCNH2 Q12809 3/20 0.40
CYP4F2 P78329 1/20 0.39
CYP4A11 Q02928 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP19A1 P11511 2/20 0.38
MTNR1A P48039 1/20 0.38
HTT P42858 2/20 0.37
LMNA P02545 1/20 0.37
HRH1 P35367 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2177576 0.84 MCHR1 (0.43) NPC1RAB9AMCHR1KCNH2LMNA
SCHEMBL2174848 0.81 MCHR1 (0.43) NPC1RAB9AMCHR1KCNH2LMNA
SCHEMBL2179048 0.79 TSHR (0.42) MCHR1KCNH2
SCHEMBL2177697 0.78 MTNR1A (0.47) ALDH1A1MTNR1AHTT
SCHEMBL2178414 0.77 TSHR (0.43) MCHR1KCNH2
SCHEMBL2175750 0.77 NPC1 (0.46) NPC1RAB9AMCHR1KCNH2ALDH1A1
SCHEMBL2177816 0.77 MCHR1 (0.46) MCHR1ALDH1A1
SCHEMBL2178661 0.76 MTNR1A (0.48) ALDH1A1MTNR1A
SCHEMBL2177993 0.75 MCHR1 (0.44) MCHR1KCNH2
SCHEMBL2177626 0.73 NPC1 (0.43) NPC1RAB9ACYP19A1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948601-A1 FAB I INHIBITOR AND PROCESS FOR PREPARING SAME Crystalgenomics, Inc. (KR) 2008-07-30 EP disclosed
WO-2007043835-A1 FAB I INHIBITOR AND PROCESS FOR PREPARING SAME CRYSTALGENOMICS, INC. (KR) 2007-04-19 WO disclosed