SCHEMBL4583744

SCHEMBL4583744

COc1ccc(C[C@@H](CO)NC(=O)OCC(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.47
LDHA P00338 1/20 0.47
ACACB O00763 1/20 0.45
PCNA P12004 1/20 0.45
ADRB1 P08588 1/20 0.44
ADRB3 P13945 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.43
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
FPR2 P25090 1/20 0.43
MMP1 P03956 2/20 0.42
SLC6A4 P31645 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073213 0.85 CYP3A4 (0.61) ALDH1A1CYP3A4MAPK1ATMCTSL
SCHEMBL4583554 0.85 CYP3A4 (0.61) ALDH1A1CYP3A4MAPK1ATMCTSL
SCHEMBL11582096 0.83 PCNA (0.55) LDHAPCNAALDH1A1CYP3A4ATM
SCHEMBL11582094 0.83 PCNA (0.55) LDHAPCNAALDH1A1CYP3A4ATM
SCHEMBL11581174 0.82 ATM (0.62) ALDH1A1CYP3A4MAPK1ATMCTSL
SCHEMBL3134015 0.82 ATM (0.62) ALDH1A1CYP3A4MAPK1ATMCTSL
SCHEMBL4356408 0.80 ACACB (0.58) LDHAACACBPCNAADRB1ADRB3
SCHEMBL14370510 0.80 ACACB (0.58) LDHAACACBPCNAADRB1ADRB3
SCHEMBL18262755 0.80 LDHA (0.58) LDHAACACBADRB1ADRB3ALDH1A1
SCHEMBL20661670 0.80 ATM (0.53) CACNA1BLDHAACACBPCNAADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed