SCHEMBL458554

SCHEMBL458554

CC(C)(C)OC(=O)Nc1cc(N2CCN(C(=O)O)CC2)c(Cl)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPY2R P49146 10/20 0.42
BACE1 P56817 2/20 0.38
MAPK8 P45983 1/20 0.38
REV1 Q9UBZ9 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
RBP4 P02753 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470197 0.90 MEN1 (0.47) BACE1MAPK8MEN1KMT2ALMNA
SCHEMBL459978 0.90 BACE1 (0.41) NPY2RBACE1MAPK8REV1LMNA
SCHEMBL12272881 0.88 ATR (0.41) NPY2RBACE1REV1KMT2ALMNA
SCHEMBL27913497 0.87 NPY2R (0.38) NPY2RBACE1MAPK8REV1MEN1
SCHEMBL459977 0.87 NPY2R (0.38) NPY2RBACE1MAPK8REV1MEN1
SCHEMBL27913478 0.83 MAPT (0.52) NPY2RMEN1KMT2ALMNAMAPK1
SCHEMBL27931713 0.82 NPY2R (0.48) NPY2RMEN1KMT2AMAPT
SCHEMBL457432 0.81 MEN1 (0.51) BACE1MAPK8MEN1KMT2ALMNA
SCHEMBL470212 0.81 MEN1 (0.51) BACE1MAPK8MEN1KMT2ALMNA
SCHEMBL463132 0.80 BACE1 (0.49) BACE1MAPK8MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103201268-B As the novel piperazine analogue of wide spectrum influenza virus medicine BRISTOL-MYERS SQUIBB CO. (US) 2015-08-12 CN disclosed
EP-2614052-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS Bristol-Myers Squibb Company (US) 2013-07-17 EP disclosed
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed