SCHEMBL470212

SCHEMBL470212

Cc1cc(Cl)c(NC(=O)OC(C)(C)C)cc1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
BACE1 P56817 2/20 0.43
MAPK8 P45983 1/20 0.43
MAPT P10636 6/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TSHR P16473 1/20 0.43
CCNK O75909 1/20 0.42
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CCND3 P30281 1/20 0.42
CDK9 P50750 1/20 0.42
CDK6 Q00534 1/20 0.42
F13A1 P00488 2/20 0.41
TGM2 P21980 2/20 0.41
TGM1 P22735 2/20 0.41
TGM3 Q08188 1/20 0.41
LMNA P02545 3/20 0.41
STS P08842 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457432 0.91 MEN1 (0.51) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL470197 0.91 MEN1 (0.47) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL470229 0.89 MEN1 (0.46) MEN1KMT2ABACE1MAPTSMN1; SMN2
SCHEMBL470227 0.87 BACE1 (0.47) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL12523337 0.84 NR1H2 (0.45) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL463132 0.83 BACE1 (0.49) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL458534 0.81 MAPT (0.58) MEN1KMT2AMAPK8MAPTSMN1; SMN2
SCHEMBL29796094 0.81 BACE1 (0.48) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL470218 0.81 BACE1 (0.48) MEN1KMT2ABACE1MAPK8MAPT
SCHEMBL458554 0.81 NPY2R (0.42) MEN1KMT2ABACE1MAPK8MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed