SCHEMBL4585884

SCHEMBL4585884

COC(=O)C(Cc1ccc2c(cnn2C(=O)O)c1)NC(=O)N1CCC(N2Cc3ccccc3NC2=O)CC1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 18/20 0.57
CYP3A4 P08684 11/20 0.57
CALCA P06881 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3595869 0.91 CALCRL (0.54) CALCRLCYP3A4CALCA
SCHEMBL3601804 0.85 CALCRL (0.53) CALCRLCYP3A4CALCA
SCHEMBL3601800 0.85 CALCRL (0.53) CALCRLCYP3A4CALCA
SCHEMBL3607821 0.84 CALCRL (0.76) CALCRLCYP3A4CALCA
SCHEMBL3607815 0.84 CALCRL (0.76) CALCRLCYP3A4CALCA
SCHEMBL3591393 0.83 CALCA (0.57) CALCRLCYP3A4CALCA
SCHEMBL3282021 0.83 CALCA (0.60) CALCRLCYP3A4CALCA
SCHEMBL3597734 0.83 CALCA (0.55) CALCRLCYP3A4CALCA
SCHEMBL3587479 0.82 CALCRL (0.60) CALCRLCYP3A4CALCA
SCHEMBL3587476 0.82 CALCRL (0.60) CALCRLCYP3A4CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100558728-C Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2009-11-11 CN disclosed
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP disclosed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP disclosed
CN-1671711-A Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2005-09-21 CN disclosed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO disclosed