SCHEMBL458643

SCHEMBL458643

Nc1nc(-c2nn(Cc3ccccc3F)c3ncccc23)nc(N)c1N(C(=O)O)C1COC1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.64
KCNH2 Q12809 1/20 0.64
GUCY1A1 Q02108 13/20 0.53
GUCY1B1 Q02153 13/20 0.53
PDE5A O76074 5/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460154 0.94 ADORA3 (0.61) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL459590 0.94 ADORA3 (0.61) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL460959 0.92 ADORA3 (0.66) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL174915 0.84 ADORA3 (0.82) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL30507540 0.84 ADORA3 (0.82) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL459275 0.84 ADORA3 (0.66) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL18496418 0.83 ADORA3 (0.81) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL5765138 0.83 ADORA3 (0.73) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL460196 0.82 ADORA3 (0.69) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL174220 0.82 ADORA3 (0.68) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012010576-A1 CARBAMATE-SUBSTITUTED DIAMINOPYRIMIDINES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-26 WO disclosed