SCHEMBL4587419

SCHEMBL4587419

CNc1ccnc2ccc(/C=C3/SC(Nc4c(Cl)cccc4Cl)=NC3=O)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CISD1 Q9NZ45 2/20 0.39
CLK1 P49759 4/20 0.38
DYRK1A Q13627 4/20 0.38
DYRK2 Q92630 3/20 0.38
DYRK1B Q9Y463 3/20 0.38
CLK2 P49760 2/20 0.38
DYRK3 O43781 2/20 0.38
CLK3 P49761 2/20 0.38
CLK4 Q9HAZ1 2/20 0.38
CSNK1E P49674 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK4 Q9NR20 1/20 0.38
PIK3CD O00329 3/20 0.38
CSNK2A2 P19784 3/20 0.38
PIK3CA P42336 3/20 0.38
PIK3CG P48736 3/20 0.38
PIK3CB P42338 2/20 0.38
MTOR P42345 2/20 0.38
PIM1 P11309 2/20 0.38
GAK O14976 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2981460 1.00 CISD1 (0.39) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2981459 1.00 CISD1 (0.39) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2993530 0.89 CLK1 (0.41) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2993535 0.89 CLK1 (0.41) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2993709 0.88 CISD1 (0.40) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2993707 0.88 CISD1 (0.40) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2991901 0.86 MEN1 (0.47) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2996253 0.86 CISD1 (0.41) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2991896 0.86 MEN1 (0.47) CISD1CLK1DYRK1ADYRK2DYRK1B
SCHEMBL2996250 0.86 CISD1 (0.41) CISD1CLK1DYRK1ADYRK2DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP claimed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP claimed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO claimed
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP disclosed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP disclosed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed