SCHEMBL4587739

SCHEMBL4587739

Cc1ccc(-c2ccc(Cl)cc2)cc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
AR P10275 4/20 0.45
S1PR1 P21453 5/20 0.44
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
ALOX5 P09917 1/20 0.39
HTT P42858 2/20 0.39
CCNE2 O96020 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
PGR P06401 1/20 0.38
KIF11 P52732 2/20 0.38
HSD11B1 P28845 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5949422 0.90 AR (0.52) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL30742957 0.88 NOTUM (0.53) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL5949403 0.88 NOTUM (0.53) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL30742956 0.88 NOTUM (0.53) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL17297890 0.84 AR (0.61) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL5936706 0.84 NOTUM (0.47) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL170669 0.84 CYP3A4 (0.46) NOTUMS1PR1HTTHSD11B1KDM4E
SCHEMBL4636314 0.82 S1PR1 (0.60) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL26375379 0.82 NOTUM (0.46) NOTUMARS1PR1PDE3BPDE3A
SCHEMBL26375434 0.82 KIF11 (0.48) NOTUMARS1PR1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377289-A4 HETEROCYCLIC COMPOUNDS FOR THERAPEUTIC USE JB CHEMICALS & PHARMACEUTICALS (IN) 2008-09-10 EP disclosed
EP-1377289-A2 HETEROCYCLIC COMPOUNDS FOR THERAPEUTIC USE J.B. Chemicals & Pharmaceuticals Ltd. (IN) 2004-01-07 EP disclosed
WO-2002074235-A2 HETEROCYCLIC COMPOUNDS FOR THERAPEUTIC USE J.B. CHEMICALS & PHARMACEUTICALS LTD (IN) 2002-09-26 WO disclosed