SCHEMBL4589004

SCHEMBL4589004

CC(C)(C)OC(=O)n1cc(-c2ccc3nc(N)n[n+]([O-])c3c2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.45
SCD O00767 1/20 0.36
GSK3B P49841 2/20 0.36
DYRK1A Q13627 2/20 0.36
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
WNT1 P04628 1/20 0.34
PIK3CA P42336 4/20 0.33
PIK3CD O00329 3/20 0.33
PI4KA P42356 3/20 0.33
PIK3CG P48736 3/20 0.33
PI4KB Q9UBF8 3/20 0.33
PIK3CB P42338 2/20 0.33
LRRK2 Q5S007 1/20 0.33
TTK P33981 1/20 0.33
LIPC P11150 1/20 0.33
GPR119 Q8TDV5 2/20 0.33
MET P08581 1/20 0.32
PIP5K1C O60331 1/20 0.32
TBK1 Q9UHD2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL780984 0.79 IDO1 (0.39) ROCK2SCD
SCHEMBL4351957 0.77 ROCK2 (0.44) ROCK2SCDGSK3BDYRK1AHSP90AA1
SCHEMBL15742917 0.75 ROCK2 (0.60) ROCK2SCDGSK3BDYRK1AWNT1
SCHEMBL23607857 0.74 ROCK2 (0.51) ROCK2SCDGSK3BDYRK1AWNT1
SCHEMBL30969365 0.74 ROCK2 (0.51) ROCK2SCDGSK3BDYRK1AWNT1
SCHEMBL559016 0.73 GSK3B (0.53) ROCK2GSK3BDYRK1AWNT1TTK
SCHEMBL4355201 0.72 ROCK2 (0.42) ROCK2SCDGSK3BDYRK1AHSP90AA1
SCHEMBL14771857 0.72 ROCK2 (0.54) ROCK2SCDGSK3BDYRK1APIK3CD
SCHEMBL31147953 0.72 ROCK2 (0.51) ROCK2SCDGSK3BDYRK1AWNT1
SCHEMBL29640785 0.72 ROCK2 (0.54) ROCK2SCDGSK3BDYRK1APIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008059259-A2 ANTICANCER COMPOUNDS WITH A BENZO ( 1, 2, 4 ) TRIAZIN-3YL-AMINE CORE SENTINEL ONCOLOGY LIMITED (GB) 2008-05-22 WO disclosed