SCHEMBL4589419

SCHEMBL4589419

COc1c(Br)ccc2ccc(=O)[nH]c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.53
CA9 Q16790 6/20 0.53
NQO2 P16083 6/20 0.38
CYP19A1 P11511 5/20 0.38
GRIN2D O15399 2/20 0.38
GRIN3B O60391 2/20 0.38
GRIN1 Q05586 2/20 0.38
GRIN2A Q12879 2/20 0.38
GRIN2B Q13224 2/20 0.38
GRIN2C Q14957 2/20 0.38
GRIN3A Q8TCU5 2/20 0.38
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 1/20 0.34
CA1 P00915 2/20 0.33
CA7 P43166 2/20 0.33
CA13 Q8N1Q1 2/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30908307 0.80 CYP19A1 (0.46) CA12CA9NQO2CYP19A1KDM4E
SCHEMBL3140886 0.76 CA12 (0.58) CA12CA9GRIN2DGRIN3BGRIN1
SCHEMBL2305754 0.74 BRD4 (0.41) NQO2CA4ALOX5APFEN1
SCHEMBL25249996 0.74 PDE3B (0.45) CA12CA9NQO2CYP19A1GRIN2D
SCHEMBL17509822 0.73 NQO2 (0.70) NQO2CYP19A1KDM4EALDH1A1HPGD
SCHEMBL29970624 0.72 CA12 (0.58) CA12CA9ALDH1A1CA1CA7
SCHEMBL21631578 0.72 CA12 (0.58) CA12CA9ALDH1A1CA1CA7
SCHEMBL4573974 0.72 CA12 (0.58) CA12CA9KDM4EALDH1A1HPGD
SCHEMBL30516741 0.71 STING1 (0.40) CA12CA9GRIN2DGRIN3BGRIN1
SCHEMBL6378203 0.71 CA12 (0.45) CA12CA9NQO2CYP19A1GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008120003-A1 SUBSTITUTED PIPERIDINES FOR USE IN THE TREATMENT OF BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2008-10-09 WO disclosed