SCHEMBL4590019

SCHEMBL4590019

O=CCCSC[CH]CCc1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
DAO P14920 3/20 0.37
IDO1 P14902 3/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
AOC3 Q16853 1/20 0.35
KCNH2 Q12809 1/20 0.35
PNMT P11086 1/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4589466 0.88 TAAR1 (0.42) TAAR1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4558176 0.88 TAAR1 (0.40) TAAR1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL30444061 0.80 TAAR1 (0.54) TAAR1DAOIDO1SLC6A2SLC6A4
SCHEMBL1338205 0.80 TAAR1 (0.54) TAAR1DAOIDO1SLC6A2SLC6A4
SCHEMBL13711753 0.74 TAAR1 (0.50) TAAR1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4589981 0.74 TAAR1 (0.41) TAAR1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4590021 0.74 CHRM2 (0.43) TAAR1DAOAOC3PNMTHTR3E
SCHEMBL3267837 0.73 TAAR1 (0.50) TAAR1DAOIDO1SLC6A2SLC6A4
SCHEMBL5541608 0.72 TAAR1 (0.48) TAAR1DAOIDO1SLC6A2SLC6A4
SCHEMBL4517362 0.72 TAAR1 (0.40) TAAR1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937656-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS BETA 2 ADRENOCEPTOR AGONISTS AstraZeneca AB (SE) 2008-07-02 EP disclosed
WO-2007027134-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS β2 ADRENOCEPTOR AGONISTS ASTRAZENECA AB (SE) 2007-03-08 WO disclosed