SCHEMBL4590227

SCHEMBL4590227

O=C(OCc1ccccc1)N1CCc2nc(N3CCNCC3)sc2C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48
SLC29A1 Q99808 1/20 0.47
DHFR P00374 1/20 0.47
KDR P35968 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TMEM97 Q5BJF2 7/20 0.43
SIGMAR1 Q99720 7/20 0.43
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GRM5 P41594 3/20 0.41
F2 P00734 1/20 0.41
F12 P00748 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19283965 0.87 MEN1 (0.47) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL19283959 0.84 GCK (0.48) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL30717385 0.83 MEN1 (0.46) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL19283878 0.82 SLC29A1 (0.47) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL9095158 0.82 MEN1 (0.54) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL3820812 0.81 DHFR (0.54) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL20509404 0.79 DHFR (0.55) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL19283880 0.79 MEN1 (0.41) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL9094028 0.78 MEN1 (0.52) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL3541178 0.77 MEN1 (0.52) MEN1KMT2AALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed