SCHEMBL4590367

SCHEMBL4590367

CC1CN(c2ccn(C3CC3)c(=O)c2)CCN1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
FAAH O00519 6/20 0.42
CHRM4 P08173 2/20 0.40
NOTUM Q6P988 1/20 0.39
CTSB P07858 2/20 0.39
CTSS P25774 2/20 0.39
CTSK P43235 2/20 0.39
CHRM2 P08172 6/20 0.38
CHRM1 P11229 5/20 0.38
SUV39H2 Q9H5I1 1/20 0.38
GRM1 Q13255 1/20 0.37
CHRM5 P08912 1/20 0.36
CHRM3 P20309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4590280 0.84 SUV39H2 (0.49) FAAHSUV39H2
SCHEMBL4590279 0.84 SUV39H2 (0.49) FAAHSUV39H2
SCHEMBL4590454 0.81 NPC1 (0.40) NPC1FAAHCHRM4CTSBCTSS
SCHEMBL27606539 0.77 FAAH (0.54) NPC1FAAHCHRM4NOTUMCTSB
SCHEMBL20139213 0.77 FAAH (0.54) NPC1FAAHCHRM4NOTUMCTSB
SCHEMBL23777734 0.76 NOTUM (0.57) NPC1FAAHNOTUM
SCHEMBL8114412 0.74 BCL2A1 (0.44)
SCHEMBL4589715 0.74 BCL2A1 (0.44)
SCHEMBL4573983 0.73 HRH3 (0.42) NPC1FAAHCHRM4CHRM2CHRM1
SCHEMBL4573827 0.72 NPC1 (0.43) NPC1FAAHCHRM4NOTUMCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed