SCHEMBL4590533

SCHEMBL4590533

COc1ccc2c(ccn2-c2ccc(Cl)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.54
ROCK1 Q13464 1/20 0.50
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
HTR2C P28335 1/20 0.46
CYP19A1 P11511 1/20 0.45
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
POLB P06746 1/20 0.43
HTR6 P50406 1/20 0.43
MIF P14174 1/20 0.43
EGFR P00533 1/20 0.42
KCNH2 Q12809 1/20 0.42
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10193341 0.90 ROCK1 (0.55) ROCK1HTR2CPDGFRBPDGFRAL3MBTL1
SCHEMBL5735721 0.84 ROCK1 (0.50) ROCK1HTR2CPDGFRBPDGFRAL3MBTL1
SCHEMBL29690879 0.84 ROCK1 (0.50) ROCK1HTR2CPDGFRBPDGFRAL3MBTL1
SCHEMBL8174904 0.84 KCNH2 (0.60) ROCK1HTR2CCYP19A1PDGFRBPDGFRA
SCHEMBL1144469 0.84 FGFR1 (0.55) ROCK1HTR2CPDGFRBPDGFRAL3MBTL1
SCHEMBL28592553 0.80 MIF (0.54) KDM4EALDH1A1HPGDSMN1; SMN2MIF
SCHEMBL5605304 0.79 ROCK1 (0.51) ROCK1HTR2CPDGFRBPDGFRAL3MBTL1
SCHEMBL6297057 0.79 MEN1 (0.46) ROCK1L3MBTL1KDM4EALDH1A1HPGD
SCHEMBL5427894 0.79 ROCK1 (0.51) ROCK1AKR1C3AKR1C2HTR2CCYP19A1
SCHEMBL21925190 0.78 ALDH1A1 (0.57) ROCK1HTR2CPDGFRBPDGFRAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107322-A1 INDOLE, BENZIMIDAZOLE OR BENZOTRIAZOLE DERIVATIVES INCLUDING A PIPERIDINE OR PIPERAZINE CORE AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed