SCHEMBL459079

SCHEMBL459079

Nc1nc(-c2nn(Cc3ccccc3F)c3ncccc23)nc(N)c1N(CC(F)(F)F)C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.68
KCNH2 Q12809 1/20 0.68
GUCY1A1 Q02108 12/20 0.54
GUCY1B1 Q02153 12/20 0.54
PDE5A O76074 6/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763523 0.92 ADORA3 (0.70) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL255819 0.91 ADORA3 (0.78) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL5765138 0.90 ADORA3 (0.73) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL7509551 0.89 ADORA3 (0.55) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL460196 0.89 ADORA3 (0.69) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL460864 0.88 ADORA3 (0.68) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL174220 0.88 ADORA3 (0.68) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL30507540 0.87 ADORA3 (0.82) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL174915 0.87 ADORA3 (0.82) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL459275 0.86 ADORA3 (0.66) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096592-B2 Bicyclic aza heterocycles, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-04 US disclosed
WO-2012010576-A1 CARBAMATE-SUBSTITUTED DIAMINOPYRIMIDINES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-26 WO disclosed