SCHEMBL4591192

SCHEMBL4591192

Cc1c(CO)nc(Nc2ccc(F)cc2)nc1N1CCc2cc(O)ccc2C1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.39
ESR2 Q92731 6/20 0.39
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
BLM P54132 1/20 0.35
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
SOS2 Q07890 1/20 0.33
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
RAD52 P43351 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
EGFR P00533 1/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6968548 0.99 ESR1 (0.39) ESR1ESR2KMT2AMEN1BLM
SCHEMBL6956974 0.89 ESR1 (0.41) ESR1ESR2KMT2AMEN1BLM
Hydrochloric Acid SCHEMBL6967452 0.88 ESR1 (0.41) ESR1ESR2KMT2AMEN1BLM
SCHEMBL4591366 0.88 KCNH3 (0.37) KMT2AMEN1BLMLMNAADRA2A
SCHEMBL7688107 0.88 ESR1 (0.39) ESR1ESR2KMT2AMEN1BLM
Hydrochloric Acid SCHEMBL6968110 0.87 KCNH3 (0.39) KMT2AMEN1BLMLMNAADRA2A
Hydrochloric Acid SCHEMBL6963712 0.83 CA1 (0.37) KMT2AMAPTLMNARAD52EGFR
SCHEMBL27417173 0.81 KMT2A (0.37) ESR1ESR2KMT2AMEN1BLM
SCHEMBL6158156 0.81 KMT2A (0.40) KMT2AMEN1BLMMAPTLMNA
Hydrochloric Acid SCHEMBL6968001 0.81 KMT2A (0.36) ESR1ESR2KMT2AMEN1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879891-A1 MUTUAL PRODRUG COMPOUNDS FOR USE AS ANTIINFLAMMATORY AGENTS WITH GASTROINTESTINAL PROTECTIVE ACTIVITY Nycomed GmbH (DE) 2008-01-23 EP claimed
WO-2006117315-A1 MUTUAL PRODRUG COMPOUNDS FOR USE AS ANTIINFLAMMATORY AGENTS WITH GASTROINTESTINAL PROTECCTIVE ACTIVITY NYCOMED GMBH (DE) 2006-11-09 WO claimed