Pyrene

Pyrene

SCHEMBL4592363

N#Cc1ccccc1C#N.c1cc2ccc3cccc4ccc(c1)c2c34

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
TSHR P16473 4/20 0.55
HSD17B10 Q99714 4/20 0.55
CYP1A2 P05177 3/20 0.55
HPGD P15428 3/20 0.55
CYP1A1 P04798 2/20 0.55
CYP1B1 Q16678 2/20 0.55
CYP3A4 P08684 2/20 0.55
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
THRB P10828 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.40
MAPK1 P28482 1/20 0.40
ATM Q13315 1/20 0.40
ERBB2 P04626 1/20 0.40
FYN P06241 1/20 0.40
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10338061 0.87 TSHR (0.50) ALDH1A1TSHRHSD17B10CYP1A2HPGD
SCHEMBL29973162 0.84 CA1 (0.50) ALDH1A1TSHRHSD17B10CYP1A2HPGD
SCHEMBL819594 0.84 CA1 (0.50) ALDH1A1TSHRHSD17B10CYP1A2HPGD
Naphthalene SCHEMBL27935169 0.84 TSHR (0.55) ALDH1A1TSHRHSD17B10CYP1A2HPGD
SCHEMBL27950969 0.82 CA1 (0.60) ALDH1A1TSHRHSD17B10CYP1A2HPGD
Hydrogen Sulfide SCHEMBL29288364 0.82 CA1 (0.48) ALDH1A1TSHRHSD17B10CYP1A2HPGD
Naphthalene SCHEMBL28320819 0.81 TSHR (0.52) ALDH1A1TSHRHSD17B10CYP1A2HPGD
SCHEMBL29352197 0.81 TSHR (0.63) ALDH1A1TSHRHSD17B10CYP1A2HPGD
SCHEMBL2818597 0.81 TSHR (0.63) ALDH1A1TSHRHSD17B10CYP1A2HPGD
Water SCHEMBL19410621 0.81 TSHR (0.63) ALDH1A1TSHRHSD17B10CYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080230715-A1 Optical Imaging KONINKLIJKE PHILIPS ELECTRONICS, N.V. (NL) 2008-09-25 US disclosed
EP-1912557-A2 OPTICAL IMAGING Philips Intellectual Property & Standards GmbH (DE) 2008-04-23 EP disclosed
WO-2007015190-A2 OPTICAL IMAGING PHILIPS INTELLECTUAL PROPERTY & STANDARDS GMBH (DE) 2007-02-08 WO disclosed