SCHEMBL4592664

SCHEMBL4592664

CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)c2cc(Br)c(Br)s2)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.56
KDM4E B2RXH2 1/20 0.53
PKM P14618 1/20 0.53
IDO1 P14902 2/20 0.49
TDO2 P48775 1/20 0.49
NAMPT P43490 2/20 0.43
CYP2C9 P11712 1/20 0.43
USP30 Q70CQ3 1/20 0.42
FPR3 P25089 1/20 0.41
FPR2 P25090 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
BRD3 Q15059 1/20 0.41
GNRHR P30968 1/20 0.41
PIK3CD O00329 1/20 0.41
KCNH2 Q12809 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
PTK2 Q05397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3447823 1.00 ACKR3 (0.56) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL3447821 1.00 ACKR3 (0.56) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL3448652 0.91 ACKR3 (0.55) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL3448647 0.91 ACKR3 (0.55) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL4592403 0.91 ACKR3 (0.55) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL3449148 0.85 ACKR3 (0.66) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL3449150 0.85 ACKR3 (0.66) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL4592230 0.85 ACKR3 (0.66) ACKR3KDM4EPKMIDO1TDO2
SCHEMBL4592619 0.84 ACKR3 (0.39) ACKR3MEN1KMT2AKCNH2CACNA1I
SCHEMBL3449326 0.80 ACKR3 (0.65) ACKR3KDM4EPKMIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877404-A2 NOVEL CYCLIC AMINES F. Hoffmann-Roche AG (CH) 2008-01-16 EP disclosed
WO-2006114401-A2 NOVEL CYCLIC AMINES F. HOFFMANN-LA ROCHE AG (CH) 2006-11-02 WO disclosed