SCHEMBL4592619

SCHEMBL4592619

O=C(NC[C@@H]1CCN(C(=O)O)C1)c1cc(Br)c(Br)s1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
GSK3B P49841 2/20 0.38
CACNA1I Q9P0X4 1/20 0.37
SMYD3 Q9H7B4 4/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KCNH2 Q12809 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592144 0.88 ACKR3 (0.40) ACKR3DRD2DRD4DRD3SMYD3
SCHEMBL3447821 0.84 ACKR3 (0.56) ACKR3MEN1KMT2ACACNA1IKCNH2
SCHEMBL3447823 0.84 ACKR3 (0.56) ACKR3MEN1KMT2ACACNA1IKCNH2
SCHEMBL4592664 0.84 ACKR3 (0.56) ACKR3MEN1KMT2ACACNA1IKCNH2
SCHEMBL4592841 0.83 GAA (0.49) ACKR3MEN1KMT2ANPSR1
SCHEMBL4592548 0.77 F10 (0.52) ACKR3
SCHEMBL4592552 0.77 F10 (0.52) ACKR3
SCHEMBL4592193 0.76 PRSS12 (0.51) KMT2A
SCHEMBL4592190 0.76 PRSS12 (0.51) KMT2A
SCHEMBL4592240 0.76 CHRNA7 (0.51) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877404-A2 NOVEL CYCLIC AMINES F. Hoffmann-Roche AG (CH) 2008-01-16 EP disclosed
WO-2006114401-A2 NOVEL CYCLIC AMINES F. HOFFMANN-LA ROCHE AG (CH) 2006-11-02 WO disclosed