SCHEMBL4593549

SCHEMBL4593549

Cc1cc(CC(CC(=O)N2CCC(N3Cc4cccc(F)c4NC3=O)CC2)C(=O)[N+]2(C3CCNCC3)CCCCC2)cc2cn[nH]c12

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 0.74
CYP3A4 P08684 2/20 0.61
CYP2D6 P10635 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5780411 0.86 CALCRL (0.67) CALCRLCYP3A4
SCHEMBL3598516 0.85 CALCRL (1.00) CALCRLCYP3A4CYP2D6
SCHEMBL4504325 0.80 CALCRL (1.00) CALCRLCYP3A4CYP2D6
SCHEMBL3598277 0.77 CALCRL (0.82) CALCRLCYP3A4CYP2D6
SCHEMBL4720735 0.77 CALCRL (0.55) CALCRL
SCHEMBL4507434 0.77 CALCRL (0.64) CALCRLCYP3A4CYP2D6
SCHEMBL4517575 0.77 CALCRL (0.75) CALCRLCYP3A4CYP2D6
SCHEMBL13756214 0.77 CALCRL (0.81) CALCRLCYP3A4CYP2D6
SCHEMBL30231296 0.76 CALCRL (1.00) CALCRLCYP3A4
SCHEMBL3607210 0.76 CALCRL (1.00) CALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP claimed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP claimed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO claimed
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP disclosed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP disclosed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO disclosed