SCHEMBL4593579

SCHEMBL4593579

CSc1nc(N)cc(-c2cc(F)c(F)c(C)c2F)n1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.36
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSP90AB1 P08238 1/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
HSP90AA1 P07900 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593134 0.82 ALDH1A1 (0.32) ALDH1A1CYP1A2GAACYP2C9CYP2C19
SCHEMBL27826457 0.76 MPL (0.45) HSP90AA1
SCHEMBL23361475 0.71 ALDH1A1 (0.47) ALDH1A1CYP1A2GAACYP2C9CYP2C19
SCHEMBL21583430 0.69 ALDH1A1 (0.55) ALDH1A1CYP1A2GAACYP2C9CYP2C19
SCHEMBL3625881 0.69 HSP90AB1 (0.46) ALDH1A1HSP90AB1NOS3NOS1NOS2
SCHEMBL8018804 0.66 KMT2A (0.49) ALDH1A1GAAHSP90AB1NOS3NOS1
SCHEMBL30718977 0.66 KMT2A (0.49) ALDH1A1GAAHSP90AB1NOS3NOS1
SCHEMBL11908093 0.66 HASPIN (0.39) CYP1A2CYP2C9CYP2C19HSP90AA1
SCHEMBL14267870 0.65 ADORA2A (0.59) ALDH1A1HSP90AB1HSP90AA1
SCHEMBL29502715 0.65 ADORA2A (0.59) ALDH1A1HSP90AB1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928842-A1 4-PHENYL-6-SUBSTITUTED-PYRIMIDINE-2-CARBONITRILE DERIVATIVES N.V. Organon (NL) 2008-06-11 EP disclosed
WO-2007039470-A1 4-PHENYL-6-SUBSTITUTED-PYRIMIDINE-2-CARBONITRILE DERIVATIVES N.V. ORGANON (NL) 2007-04-12 WO disclosed