SCHEMBL4594256

SCHEMBL4594256

Oc1ccc2oc(NC3CCNCC3)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.50
FAAH O00519 8/20 0.48
PIK3CA P42336 2/20 0.42
ESR1 P03372 4/20 0.42
ESR2 Q92731 4/20 0.42
PIK3CB P42338 1/20 0.40
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL1121793 0.99 HDAC6 (0.49) HDAC6FAAHPIK3CAESR1ESR2
Hydrochloric Acid SCHEMBL1121658 0.99 HDAC6 (0.49) HDAC6FAAHPIK3CAESR1ESR2
SCHEMBL14867048 0.90 HDAC6 (0.55) HDAC6FAAHPIK3CAESR1ESR2
SCHEMBL13543026 0.84 SSTR5 (0.48) HDAC6FAAH
SCHEMBL13543034 0.84 HDAC6 (0.47) HDAC6FAAHPIK3CA
Hydrochloric Acid SCHEMBL4947954 0.83 HDAC6 (0.46) HDAC6FAAHPIK3CA
Hydrochloric Acid SCHEMBL27695367 0.83 HDAC6 (0.46) HDAC6FAAHPIK3CA
Bromide SCHEMBL3570502 0.83 SSTR5 (0.48) HDAC6FAAH
SCHEMBL1121922 0.82 FAAH (0.52) HDAC6FAAHPIK3CA
SCHEMBL13543033 0.81 SSTR5 (0.52) HDAC6FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101253171-B Benzooxazole, oxazolopyridine, benzothiazole and thiazolopyridine derivatives HOFFMANN LA ROCHE 2011-06-15 CN disclosed
CN-101253171-A Benzooxazole, oxazolopyridine, benzothiazole and thiazolopyridine derivatives HOFFMANN LA ROCHE (CH) 2008-08-27 CN disclosed
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP disclosed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO disclosed