SCHEMBL4595035

SCHEMBL4595035

N#Cc1ccc(N(CCCC(=O)N2CCOCC2)CC(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.46
PGR P06401 1/20 0.46
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
MLYCD O95822 9/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
CETP P11597 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
POLB P06746 1/20 0.36
FKBP1A P62942 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595452 0.91 AR (0.48) ARPGRCETP
SCHEMBL4595549 0.90 AR (0.47) ARPGRALDH1A1HPGDKDM4E
SCHEMBL4619274 0.89 AR (0.46) ARPGRCETP
SCHEMBL4595143 0.85 AR (0.44) ARPGR
SCHEMBL4594140 0.77 AR (0.66) ARPGRALDH1A1HPGDKDM4E
SCHEMBL3039891 0.77 AR (0.52) ARPGR
SCHEMBL4595030 0.76 AR (0.56) ARPGRALDH1A1HPGDKDM4E
Trifluoroacetic Acid SCHEMBL3419464 0.75 AR (0.48) ARPGR
SCHEMBL3060320 0.74 AR (0.53) ARPGR
SCHEMBL3048408 0.74 AR (0.54) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871379-A2 CYANOARYLAMINES Smithkline Beecham Corporation (US) 2008-01-02 EP claimed
WO-2006113552-A2 CYANOARYLAMINES SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO claimed
EP-1871379-A2 CYANOARYLAMINES Smithkline Beecham Corporation (US) 2008-01-02 EP disclosed
WO-2006113552-A2 CYANOARYLAMINES SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed