SCHEMBL4595143

SCHEMBL4595143

N#Cc1ccc(N(CCCC(=O)N2CCSC2)CC(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.44
PGR P06401 2/20 0.44
DPP4 P27487 8/20 0.38
DPP7 Q9UHL4 3/20 0.38
S1PR1 P21453 1/20 0.36
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4619274 0.94 AR (0.46) ARPGRS1PR1RXRARXRB
SCHEMBL4595452 0.88 AR (0.48) ARPGRS1PR1RXRARXRB
SCHEMBL4595549 0.87 AR (0.47) ARPGRS1PR1RXRARXRB
SCHEMBL4595035 0.85 AR (0.46) ARPGR
SCHEMBL4904337 0.76 AR (0.54) ARPGRDPP4DPP7S1PR1
SCHEMBL3039891 0.75 AR (0.52) ARPGRRXRARXRBRXRG
Trifluoroacetic Acid SCHEMBL3419464 0.74 AR (0.48) ARPGRS1PR1RXRARXRB
SCHEMBL4595496 0.74 AR (0.66) ARPGRS1PR1RXRARXRB
SCHEMBL3060320 0.73 AR (0.53) ARPGR
SCHEMBL3048408 0.73 AR (0.54) ARPGRRXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871379-A2 CYANOARYLAMINES Smithkline Beecham Corporation (US) 2008-01-02 EP claimed
WO-2006113552-A2 CYANOARYLAMINES SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO claimed
EP-1871379-A2 CYANOARYLAMINES Smithkline Beecham Corporation (US) 2008-01-02 EP disclosed
WO-2006113552-A2 CYANOARYLAMINES SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed