SCHEMBL4595068

SCHEMBL4595068

C=CC(=O)OC(CC)O[Si](C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 8/20 0.40
HPGD P15428 1/20 0.40
ALDH1A1 P00352 4/20 0.35
TP53 P04637 2/20 0.35
HIF1A Q16665 2/20 0.35
CYP3A4 P08684 1/20 0.35
HSD17B10 Q99714 1/20 0.35
THRB P10828 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11803428 0.90 TSHR (0.36) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL4596155 0.86 TSHR (0.42) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL27778925 0.86 TSHR (0.35) TSHRHPGD
SCHEMBL2229573 0.85 TSHR (0.37) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL1138627 0.84 TSHR (0.45) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL8863672 0.84 TSHR (0.36) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL5835078 0.82 TSHR (0.35) TSHRHPGD
SCHEMBL27997405 0.81 TSHR (0.42) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL28006718 0.81 TSHR (0.34) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL28162731 0.81 TSHR (0.34) TSHRHPGDALDH1A1TP53HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137727-B1 AQUEOUS COATING COMPOSITIONS DU PONT (US) 2008-01-09 EP disclosed
EP-1619225-A2 Aqueous pigment dispersion E.I.Du pont de nemours and company (US) 2006-01-25 EP disclosed
EP-0996689-B1 PIGMENT DISPERSIONS CONTAINING HYDROXYLATED AB-BLOCK POLYMER DISPERSANT DU PONT (US) 2002-12-18 EP disclosed
US-6306521-B1 SUBSTRATE COATED WITH DRIED, CURED LAYER OF COMPOSITION OF ORGANIC LIQUID CARRIER, FILM FORMING BINDER AND PIGMENT DISPERSION, WHEREIN PIGMENT DISPERSION COMPRISES DISPERSED PIGMENT, CARRIER LIQUID AND AB-BLOCK POLYMER DISPERSANT E. I. DU PONT DE NEMOURS AND COMPANY 2001-10-23 US disclosed
EP-1137727-A1 AQUEOUS COATING COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2001-10-04 EP disclosed
US-6204319-B1 AB BLOCK COPOLYMER PIGMENT DISPERSANT RESIN OF AN A BLOCK OF A HYDROPHOBIC POLYMER HAVING AMINE GROUPS; AND A B BLOCK OF A HYDROPHILIC POLYMER HAVING HYDROXYL GROUPS AND CARBOXYL GROUPS E.I. DU PONT DE NEMOURS AND COMPANY 2001-03-20 US disclosed
US-6187854-B1 WEATHERPROOF COATINGS E. I. DU PONT DE NEMOURS AND COMPANY 2001-02-13 US disclosed
WO-2000026308-A1 AQUEOUS COATING COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2000-05-11 WO disclosed
EP-0996689-A1 PIGMENT DISPERSIONS CONTAINING HYDROXYLATED AB-BLOCK POLYMER DISPERSANT E.I. DU PONT DE NEMOURS AND COMPANY (US) 2000-05-03 EP disclosed
WO-1999003938-A1 PIGMENT DISPERSIONS CONTAINING HYDROXYLATED AB-BLOCK POLYMER DISPERSANT E.I. DU PONT DE NEMOURS AND COMPANY (US) 1999-01-28 WO disclosed
US-5859113-A COATINGS; POLYMER A SEGMENT CONSISTS OF POLYMERIZED GLYCIDYL (METH)ACRYLATE REACTED WITH AN ACID; POLYMER B SEGMENT CONTAINS REACTIVE HYDROXY ALKYL (METH)ACRYLATE MONOMERS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1999-01-12 US disclosed
US-5658988-A ONE-PACKAGE; AUTOMOBILE FINISHES KANSAI PAINT CO., LTD. (JP) 1997-08-19 US disclosed
US-3935342-A POLYMERIZATION WITH AN UNSATURATED SILYL MONOMER MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-01-27 US disclosed