SCHEMBL4596336

SCHEMBL4596336

O=C1c2ccccc2C(=O)N1CC1Cc2cc(F)cc(-c3c(Cl)cccc3Cl)c2O1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.62
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2C9 P11712 2/20 0.39
MIF P14174 1/20 0.39
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
RECQL P46063 1/20 0.36
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
KDM4E B2RXH2 1/20 0.34
RAB9A P51151 1/20 0.34
DRD2 P14416 2/20 0.34
DRD4 P21917 2/20 0.34
DRD3 P35462 2/20 0.34
PRKAB2 O43741 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4234302 1.00 AQP1 (0.62) AQP1CYP1A2CYP2C19CYP2C9MIF
SCHEMBL3344458 0.83 AQP1 (0.44) AQP1CYP1A2CYP2C19CYP2C9MIF
SCHEMBL5361629 0.83 AQP1 (0.44) AQP1CYP1A2CYP2C19CYP2C9MIF
SCHEMBL5361633 0.83 AQP1 (0.44) AQP1CYP1A2CYP2C19CYP2C9MIF
SCHEMBL4226488 0.81 AQP1 (0.65) AQP1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL28393554 0.81 CYP2C9 (0.43) AQP1CYP1A2CYP2C19CYP2C9MIF
SCHEMBL13306783 0.81 AQP1 (0.42) AQP1CYP1A2CYP2C19CYP2C9MIF
SCHEMBL4226184 0.81 AQP1 (0.64) AQP1ALDH1A1KDM4EPRKAB2PRKAG1
SCHEMBL4620582 0.80 AQP1 (0.63) AQP1TSHR
SCHEMBL4220568 0.79 AQP1 (0.72) AQP1PRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed