SCHEMBL4596664

SCHEMBL4596664

O=C(O)NCC1Cc2cc(F)cc(-c3ccccc3Cl)c2O1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.57
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
LMNA P02545 4/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
KDM4E B2RXH2 1/20 0.36
RECQL P46063 1/20 0.36
EZH2 Q15910 1/20 0.35
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4961651 0.90 AQP1 (0.59) AQP1NPC1RAB9AHPGDALDH1A1
SCHEMBL4230839 0.89 AQP1 (0.72) AQP1HPGDALDH1A1TSHRLMNA
SCHEMBL4597134 0.89 AQP1 (0.51) AQP1HPGDALDH1A1TSHRLMNA
SCHEMBL4220360 0.85 AQP1 (0.43) AQP1NPC1RAB9AHPGDALDH1A1
SCHEMBL4231359 0.85 AQP1 (0.45) AQP1HPGDALDH1A1LMNAKDM4E
SCHEMBL4230165 0.85 AQP1 (0.69) AQP1HPGDALDH1A1TSHRLMNA
SCHEMBL4224838 0.84 AQP1 (0.79) AQP1CHRM2CHRM1CHRM3CYP3A4
SCHEMBL4224840 0.84 AQP1 (0.79) AQP1CHRM2CHRM1CHRM3CYP3A4
SCHEMBL4963332 0.81 AQP1 (0.50) AQP1ALDH1A1TSHRLMNACYP3A4
SCHEMBL4963338 0.81 AQP1 (0.50) AQP1ALDH1A1TSHRLMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed