Levamfetamine

Levamfetamine

SCHEMBL4596702

C[C@@H](N)Cc1ccccc1.NC(CC(=O)O)C(=O)O

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC18A2SLC6A2SLC6A3

The experimentally established mechanism targets of Levamfetamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 2/20 0.63
SLC6A3 known ✓ Q01959 1/20 0.63
TAAR1 Q96RJ0 2/20 0.63
SLC6A4 P31645 2/20 0.63
MAOA P21397 1/20 0.63
SIGMAR1 Q99720 1/20 0.63
CYP2A6 P11509 1/20 0.63
ADORA2A P29274 1/20 0.63
ADORA1 P30542 1/20 0.63
ALPI P09923 1/20 0.62
PKM P14618 1/20 0.62
PTGS1 P23219 1/20 0.62
XIAP P98170 1/20 0.62
SLC7A5 Q01650 1/20 0.62
SLC1A3 P43003 2/20 0.58
SLC1A2 P43004 2/20 0.58
SLC1A1 P43005 2/20 0.58
CPA1 P15085 2/20 0.54
CPB1 P15086 1/20 0.54
CPA3 P15088 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dextroamphetamine SCHEMBL3681578 1.00 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1030967 1.00 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1030966 1.00 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL19285614 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1005247 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL19285616 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL30336931 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Levamfetamine SCHEMBL30083110 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Dextroamphetamine SCHEMBL21158800 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1005248 0.98 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9713592-B2 Matrix-based pulse release pharmaceutical formulation MALLINCKRODT LLC (US) 2017-07-25 US claimed
EP-1874274-A2 MATRIX-BASED PULSE RELEASE PHARMACEUTICAL FORMULATION MALLINCKRODT INC. (US) 2008-01-09 EP claimed
WO-2006107593-A2 MATRIX-BASED PULSE RELEASE PHARMACEUTICAL FORMULATION MALLINCKRODT INC. (US) 2006-10-12 WO claimed
EP-1874274-A2 MATRIX-BASED PULSE RELEASE PHARMACEUTICAL FORMULATION MALLINCKRODT INC. (US) 2008-01-09 EP disclosed
WO-2006107593-A2 MATRIX-BASED PULSE RELEASE PHARMACEUTICAL FORMULATION MALLINCKRODT INC. (US) 2006-10-12 WO disclosed