Amphetamine

Amphetamine

SCHEMBL1005248

CC(N)Cc1ccccc1.N[C@@H](CC(=O)O)C(=O)O.O

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC6A2SLC6A3

The experimentally established mechanism targets of Amphetamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 2/20 0.61
SLC6A3 known ✓ Q01959 1/20 0.61
TAAR1 Q96RJ0 2/20 0.61
SLC6A4 P31645 2/20 0.61
MAOA P21397 1/20 0.61
SIGMAR1 Q99720 1/20 0.61
CYP2A6 P11509 1/20 0.61
ADORA2A P29274 1/20 0.61
ADORA1 P30542 1/20 0.61
ALPI P09923 1/20 0.61
PKM P14618 1/20 0.61
PTGS1 P23219 1/20 0.61
XIAP P98170 1/20 0.61
SLC7A5 Q01650 1/20 0.61
SLC1A3 P43003 2/20 0.57
SLC1A2 P43004 2/20 0.57
SLC1A1 P43005 2/20 0.57
CPA1 P15085 2/20 0.53
CPB1 P15086 1/20 0.53
CPA3 P15088 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amphetamine SCHEMBL19285616 1.00 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL30336931 1.00 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Dextroamphetamine SCHEMBL21158800 1.00 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL19285614 1.00 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1005247 1.00 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Levamfetamine SCHEMBL30083110 1.00 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1030966 0.98 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3
Levamfetamine SCHEMBL4596702 0.98 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3
Dextroamphetamine SCHEMBL3681578 0.98 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1030967 0.98 SLC6A2 (0.63) SLC6A2TAAR1SLC6A4MAOASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 231 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12544385-B2 Combination drug therapies for CNS disorders JAVED MOHAMMAD (US) 2026-02-10 US claimed
US-20260027043-A1 EXTENDED RELEASE AMPHETAMINE TABLETS TRIS PHARMA INC (US) 2026-01-29 US claimed
US-12208068-B2 Amphetamine controlled release, prodrug, and abuse-deterrent dosage forms Pharmapotheca A Inc. (US) 2025-01-28 US claimed
EP-3638211-B1 DELAYED SUSTAINED RELEASE PHARMACEUTICAL COMPOSITIONS SpecGx LLC (US) 2023-11-29 EP claimed
US-20230321010-A1 Amphetamine Controlled Release, Prodrug, and Abuse-deterrent Dosage Forms CHEMAPOTHECA, LLC (US) 2023-10-12 US claimed
US-11717498-B2 Methods of treatment using amphetamine controlled release, prodrug, and abuse deterrent dosage forms Pharmapotheca A, Inc. (US) 2023-08-08 US claimed
US-20230105795-A1 COMBINATION DRUG THERAPIES FOR CNS DISORDERS JAVED MOHAMMAD (US) 2023-04-06 US claimed
EP-4096508-A1 COMBINATION DRUG THERAPIES FOR CNS DISORDERS Javed, Mohammad (US) 2022-12-07 EP claimed
US-11123310-B2 Amphetamine controlled release, prodrug, and abuse-deterrent dosage forms PHARMAPOTHECA, LLC (US) 2021-09-21 US claimed
WO-2021154631-A1 COMBINATION DRUG THERAPIES FOR CNS DISORDERS JAVED MOHAMMAD (US) 2021-08-05 WO claimed
EP-2023900-A1 CONTROLLED DOSE DRUG DELIVERY SYSTEM Shire LLC (US) 2009-02-18 EP claimed
WO-2007133203-A1 CONTROLLED DOSE DRUG DELIVERY SYSTEM SHIRE LLC (US) 2007-11-22 WO claimed
US-20070264323-A1 CONTROLLED DOSE DRUG DELIVERY SYSTEM SHIRE LLC (US) 2007-11-15 US claimed
US-20060204575-A1 Amphetamine formulations ACTAVIS GROUP PTC EHF 2006-09-14 US claimed
US-20050158384-A1 Sustained release delivery of amphetamine salts SHIRE LLC 2005-07-21 US claimed
EP-1542660-A1 SUSTAINED RELEASED DELIVERY OF AMPHETAMINE SALTS Shire Laboratories Inc. (US) 2005-06-22 EP claimed
WO-2005044238-A1 MODIFIED RELEASE SOLID DOSAGE FORM OF AMPHETAMINE SALTS RANBAXY LABORATORIES LIMITED (IN) 2005-05-19 WO claimed
WO-2004028509-A1 SUSTAINED RELEASED DELIVERY OF AMPHETAMINE SALTS SHIRE LABORATORIES, INC. (US) 2004-04-08 WO claimed
US-20040059002-A1 Sustained release delivery of amphetamine salts SHIRE LABORATORIES, INC. 2004-03-25 US claimed
US-6605300-B1 For treatment of ADHD SHIRE LABORATORIES, INC. 2003-08-12 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12544385-B2 Combination drug therapies for CNS disorders SLC6A3, SLC6A2, SLC18A2 SLC6A2 2/4885SLC6A3 1/4885TAAR1 63/4885
US-11123310-B2 Amphetamine controlled release, prodrug, and abuse-deterrent dosage forms SLC6A3, CES2, SLC6A2 SLC6A2 3/4885SLC6A3 1/4885TAAR1 52/4885
US-11717498-B2 Methods of treatment using amphetamine controlled release, prodrug, and abuse deterrent dosage forms SLC6A3, SLC6A2, CES2 SLC6A2 2/4885SLC6A3 1/4885TAAR1 51/4885
US-20260027043-A1 EXTENDED RELEASE AMPHETAMINE TABLETS SLC6A3, SLC6A2, SLC6A4 SLC6A2 2/4885SLC6A3 1/4885TAAR1 238/4885
US-20230321010-A1 Amphetamine Controlled Release, Prodrug, and Abuse-deterrent Dosage Forms SLC6A3, CES2, SLC6A2 SLC6A2 3/4885SLC6A3 1/4885TAAR1 37/4885
US-12208068-B2 Amphetamine controlled release, prodrug, and abuse-deterrent dosage forms SLC6A3, CES2, SLC6A2 SLC6A2 3/4885SLC6A3 1/4885TAAR1 37/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.