SCHEMBL4596884

SCHEMBL4596884

O=C1CCNc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=C1Nc2ccc(-c3ccc(C(F)(F)F)cc3)cc2CC1O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 9/20 0.59
TDP2 O95551 1/20 0.41
AKT1 P31749 2/20 0.40
PDE3B Q13370 3/20 0.39
PDE3A Q14432 3/20 0.39
CYP1A2 P05177 2/20 0.38
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
CYP2C9 P11712 1/20 0.38
TBXAS1 P24557 1/20 0.38
CDK1 P06493 1/20 0.38
KIT P10721 1/20 0.38
CDK2 P24941 1/20 0.38
KDR P35968 1/20 0.38
PARP10 Q53GL7 1/20 0.36
PARP11 Q9NR21 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
CHRNB2 P17787 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596144 0.87 KIF11 (0.60) KIF11TDP2AKT1PDE3BPDE3A
SCHEMBL4596333 0.84 KIF11 (0.68) KIF11TDP2PDE3BPDE3ACYP1A2
SCHEMBL4596504 0.81 KIF11 (0.61) KIF11TDP2AKT1PDE3BPDE3A
SCHEMBL1396616 0.76 KIF11 (1.00) KIF11TDP2AKT1PDE3BPDE3A
SCHEMBL4596892 0.73 KIF11 (0.42) KIF11TDP2PDE3BPDE3ACYP1A2
SCHEMBL4888861 0.72 KIF11 (0.86) KIF11TDP2AKT1PDE3BPDE3A
SCHEMBL4888035 0.72 KIF11 (0.86) KIF11TDP2AKT1PDE3BPDE3A
SCHEMBL4891219 0.72 KIF11 (0.56) KIF11TDP2AKT1PDE3BPDE3A
SCHEMBL4596404 0.72 KIF11 (0.44) KIF11CYP11B1CYP11B2
SCHEMBL4594888 0.72 KIF11 (0.56) KIF11TDP2AKT1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP claimed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO claimed
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed