SCHEMBL4597328

SCHEMBL4597328

NC(=O)c1cccc(CNc2c(Nc3ccc4nc[nH]c4c3)c(=O)c2=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 4/20 0.47
AURKA O14965 2/20 0.47
NAMPT P43490 1/20 0.46
RPS6KB1 P23443 3/20 0.45
CHEK1 O14757 2/20 0.45
DAPK3 O43293 2/20 0.45
ROCK2 O75116 2/20 0.45
CHEK2 O96017 2/20 0.45
PRKACA P17612 2/20 0.45
AKT1 P31749 2/20 0.45
AKT2 P31751 2/20 0.45
CLK2 P49760 2/20 0.45
GSK3B P49841 2/20 0.45
RPS6KA3 P51812 2/20 0.45
PRKAA1 Q13131 2/20 0.45
PRKG2 Q13237 2/20 0.45
ROCK1 Q13464 2/20 0.45
PRKG1 Q13976 2/20 0.45
PKN2 Q16513 2/20 0.45
CDC42BPA Q5VT25 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4909000 0.92 AURKB (0.47) AURKBAURKANAMPTRPS6KB1CHEK1
SCHEMBL4596911 0.87 NAMPT (0.47) AURKBAURKANAMPTRPS6KB1CHEK1
SCHEMBL14066719 0.84 IP6K1 (0.55) AURKBNAMPTRPS6KB1CHEK1DAPK3
SCHEMBL4925323 0.83 ROCK2 (0.48) AURKBNAMPTRPS6KB1CHEK1DAPK3
SCHEMBL4907453 0.82 ROCK2 (0.54) AURKBAURKANAMPTRPS6KB1CHEK1
SCHEMBL4908067 0.81 GSK3B (0.44) AURKBAURKARPS6KB1CHEK1DAPK3
SCHEMBL4907508 0.81 QPCT (0.46) AURKBNAMPTRPS6KB1CHEK1DAPK3
SCHEMBL4598622 0.80 QPCT (0.50) AURKBNAMPTRPS6KB1CHEK1DAPK3
SCHEMBL4598175 0.80 MAPK1 (0.47) AURKBAURKANAMPTRPS6KB1CHEK1
SCHEMBL4905319 0.79 QPCT (0.46) AURKBNAMPTRPS6KB1CHEK1DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed