SCHEMBL4597349

SCHEMBL4597349

CC1CN(Cc2ccc(CCC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CC(C)N1C(=O)OC(C)(C)C

nearest known ligand 0.70

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MLNR O43193 17/20 0.70
CYP3A4 P08684 8/20 0.57
ALDH1A1 P00352 2/20 0.46
CYP2D6 P10635 2/20 0.45
GHSR Q92847 1/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1703823 1.00 MLNR (0.70) MLNRCYP3A4ALDH1A1CYP2D6GHSR
SCHEMBL4183557 0.88 MLNR (0.77) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL1704816 0.87 MLNR (0.74) MLNRCYP3A4ALDH1A1CYP2D6GHSR
SCHEMBL1704684 0.85 MLNR (0.71) MLNRCYP3A4ALDH1A1CYP2D6GHSR
SCHEMBL1704619 0.82 MLNR (1.00) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL4185674 0.82 MLNR (0.73) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL5125893 0.80 MLNR (0.74) MLNRCYP3A4CYP2D6GHSR
SCHEMBL11967642 0.79 MLNR (0.66) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL1703977 0.79 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704131 0.79 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907374-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-04-09 EP disclosed
WO-2007012479-A2 BENZYLPIPERAZINE DERIVATES AND THEIR MEDICAL USE GLAXO GROUP LIMITED (GB) 2007-02-01 WO disclosed