SCHEMBL4597553

SCHEMBL4597553

COC(=O)Cc1ccc(CN2CC[N+](C(=O)[O-])(C(C)(C)C)[C@@H](C)C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 2/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
MMP9 P14780 1/20 0.36
NPC1 O15118 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 1/20 0.35
EPHX2 P34913 1/20 0.35
LIPE Q05469 1/20 0.35
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3914828 0.86 DRD2 (0.39) SMN1; SMN2RAB9AALDH1A1DRD2DRD4
SCHEMBL3921081 0.85 DRD2 (0.40) ALDH1A1DRD2DRD4SIGMAR1LMNA
SCHEMBL3912115 0.85 DRD2 (0.40) ALDH1A1DRD2DRD4SIGMAR1LMNA
SCHEMBL3914146 0.83 KDM4E (0.46) SMN1; SMN2RAB9AALDH1A1NPC1SIGMAR1
SCHEMBL3912803 0.83 KDM4E (0.46) SMN1; SMN2RAB9AALDH1A1NPC1SIGMAR1
SCHEMBL3924819 0.79 CNR2 (0.37) DRD2DRD4
SCHEMBL3936339 0.79 EPHX2 (0.37) RAB9AALDH1A1DRD2DRD4EPHX2
SCHEMBL3925482 0.78 DPP4 (0.38) RAB9AALDH1A1DRD2DRD4EPHX2
SCHEMBL3936344 0.76 KDM4E (0.38) SMN1; SMN2RAB9AALDH1A1DRD2DRD4
SCHEMBL3933234 0.74 DRD2 (0.35) SMN1; SMN2ALDH1A1DRD2DRD4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907374-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-04-09 EP disclosed
WO-2007012479-A2 BENZYLPIPERAZINE DERIVATES AND THEIR MEDICAL USE GLAXO GROUP LIMITED (GB) 2007-02-01 WO disclosed