SCHEMBL4597800

SCHEMBL4597800

Clc1cc[c]cn1.O=Cc1c[nH]c2ncccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.68
CHEK1 O14757 2/20 0.40
CDK9 P50750 5/20 0.40
CDC7 O00311 4/20 0.40
DAPK3 O43293 3/20 0.40
MAP4K4 O95819 3/20 0.40
PIM1 P11309 3/20 0.40
PRKACA P17612 3/20 0.40
CLK2 P49760 3/20 0.40
GSK3B P49841 3/20 0.40
CDK7 P50613 3/20 0.40
PRKX P51817 3/20 0.40
CDK5 Q00535 3/20 0.40
DYRK1A Q13627 3/20 0.40
CLK4 Q9HAZ1 3/20 0.40
FLT3 P36888 2/20 0.40
CDK8 P49336 2/20 0.40
PKN2 Q16513 2/20 0.40
MINK1 Q8N4C8 2/20 0.40
HIPK2 Q9H2X6 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257134 0.82 KMT2A (1.00) KMT2ACHEK1CDK9CDC7LRRK2
SCHEMBL29768777 0.82 KMT2A (1.00) KMT2ACHEK1CDK9CDC7LRRK2
SCHEMBL29768778 0.82 KMT2A (1.00) KMT2ACHEK1CDK9CDC7LRRK2
Alcohol SCHEMBL27754790 0.74 KMT2A (0.82) KMT2ACHEK1CDK9CDC7LRRK2
SCHEMBL15331290 0.68 KMT2A (0.71) KMT2ACHEK1CDK9LRRK2AXL
SCHEMBL15331287 0.68 KMT2A (0.71) KMT2ACHEK1CDK9LRRK2AXL
SCHEMBL857987 0.68 KMT2A (0.52) KMT2ACHEK1CDK9CDC7DAPK3
SCHEMBL858196 0.68 KMT2A (0.52) KMT2ACHEK1CDK9CDC7DAPK3
SCHEMBL73686 0.67
SCHEMBL1772824 0.67 KMT2A (0.69) KMT2ACHEK1CDK9CDC7MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885723-A2 PYRROLO[2,3-B]PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2008-02-13 EP disclosed
WO-2007013896-A2 PYRROL (2,3-B) PYRIDINE DERIVATIVES PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-02-01 WO disclosed