SCHEMBL4597813

SCHEMBL4597813

Cn1ncc2c1CN(C(=O)Nc1ccc(Cl)cc1)C2C(=O)Nc1ccc(-n2ccncc2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F10 P00742 17/20 0.38
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34
TRPV1 Q8NER1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14097939 1.00 F10 (0.38) F10NPC1CYP1A2CYP2D6CYP2C19
SCHEMBL14138802 0.92 F10 (0.36) F10NPC1CYP2C19RAB9A
SCHEMBL4598104 0.90 F10 (0.48) F10
SCHEMBL4598445 0.90 F10 (0.48) F10
SCHEMBL14627677 0.89 F10 (0.34) F10
SCHEMBL4599259 0.89 F10 (0.51) F10
SCHEMBL4604029 0.83 F10 (0.42) F10
SCHEMBL4606187 0.83 F10 (0.42) F10
SCHEMBL14138393 0.82 F10 (0.41) F10
SCHEMBL14627717 0.80 F10 (0.40) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907388-A1 NOVEL HETEROARYL FUSED CYCLIC AMINES F. Hoffmann-Roche AG (CH) 2008-04-09 EP disclosed
WO-2007009883-A1 NOVEL HETEROARYL FUSED CYCLIC AMINES F. HOFFMANN-LA ROCHE AG (CH) 2007-01-25 WO disclosed