SCHEMBL459787

SCHEMBL459787

Fc1cncc(-c2nc3ccc(F)cc3n2C2CC2)c1

nearest known ligand 0.79

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 20/20 0.79
CYP11B1 P15538 17/20 0.79
CYP19A1 P11511 2/20 0.74
ADRA2B P18089 2/20 0.74
ADRB1 P08588 1/20 0.73
ADRA2A P08913 1/20 0.73
ADRA2C P18825 1/20 0.73
HTR2C P28335 1/20 0.73
HTR2B P41595 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896719 0.90 CYP11B2 (0.74) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL10175363 0.89 CYP11B2 (0.71) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL10175136 0.89 CYP11B2 (0.70) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL20337618 0.88 CYP11B2 (1.00) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17896594 0.88 CYP11B2 (0.78) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17896605 0.86 CYP11B2 (0.71) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL10175336 0.86 CYP11B2 (0.76) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL459353 0.85 CYP11B2 (1.00) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL460209 0.85 CYP11B2 (1.00) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
Msd-Cyp11B2 SCHEMBL31477726 0.85 CYP11B2 (1.00) CYP11B2CYP11B1CYP19A1ADRA2BADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP claimed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO claimed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed