SCHEMBL4598328

SCHEMBL4598328

Cc1cc(Nc2c(NCc3cccc(O)c3)c(=O)c2=O)cc2[nH]cnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.43
RPS6KB1 P23443 7/20 0.43
AURKB Q96GD4 7/20 0.43
ROCK1 Q13464 7/20 0.43
PRKG1 Q13976 7/20 0.43
CHEK2 O96017 6/20 0.43
PRKACA P17612 6/20 0.43
RPS6KA3 P51812 6/20 0.43
PKN2 Q16513 6/20 0.43
CDC42BPA Q5VT25 6/20 0.43
HIPK4 Q8NE63 6/20 0.43
GSK3A P49840 6/20 0.43
ROCK2 O75116 5/20 0.43
AKT1 P31749 5/20 0.43
CSNK1G3 Q9Y6M4 5/20 0.43
NEK4 P51957 4/20 0.43
MATK P42679 1/20 0.43
CLK4 Q9HAZ1 7/20 0.42
CHEK1 O14757 5/20 0.42
MKNK2 Q9HBH9 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598263 0.88 AURKB (0.43) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4906437 0.84 RPS6KB1 (0.43) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4596911 0.82 NAMPT (0.47) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4911057 0.81 CHEK2 (0.50) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4905587 0.80 ROCK1 (0.48) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4905562 0.80 KDR (0.44) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4598858 0.78 GSK3B (0.39) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4598166 0.77 RPS6KB1 (0.37) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL4917069 0.77 EGFR (0.50) GSK3BRPS6KB1AURKBROCK1PRKG1
SCHEMBL1228940 0.76 RPS6KB1 (0.44) GSK3BRPS6KB1AURKBROCK1PRKG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed