SCHEMBL4598263

SCHEMBL4598263

O=c1c(NCc2cccc(O)c2)c(Nc2cc(Cl)c3nc[nH]c3c2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 7/20 0.43
RPS6KB1 P23443 6/20 0.43
CHEK2 O96017 6/20 0.43
PRKACA P17612 6/20 0.43
RPS6KA3 P51812 6/20 0.43
ROCK1 Q13464 6/20 0.43
CDC42BPA Q5VT25 6/20 0.43
AKT1 P31749 5/20 0.43
GSK3B P49841 5/20 0.43
PRKG1 Q13976 5/20 0.43
PKN2 Q16513 5/20 0.43
HIPK4 Q8NE63 5/20 0.43
PRKAA1 Q13131 5/20 0.43
ROCK2 O75116 5/20 0.43
GSK3A P49840 5/20 0.43
CHEK1 O14757 4/20 0.43
PRKG2 Q13237 4/20 0.43
CLK4 Q9HAZ1 4/20 0.43
MKNK2 Q9HBH9 4/20 0.43
SGK2 Q9HBY8 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598328 0.88 GSK3B (0.43) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4908175 0.84 RPS6KB1 (0.43) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4596911 0.82 NAMPT (0.47) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4905587 0.80 ROCK1 (0.48) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4919796 0.77 GSK3B (0.48) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4598858 0.76 GSK3B (0.39) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4598401 0.76 KDR (0.47) AURKBRPS6KB1ABL1KDRAURKA
SCHEMBL4898767 0.76 RPS6KB1 (0.40) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4906437 0.76 RPS6KB1 (0.43) AURKBRPS6KB1CHEK2PRKACARPS6KA3
SCHEMBL4898803 0.74 ROCK2 (0.50) AURKBRPS6KB1CHEK2PRKACARPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed