SCHEMBL4598959

SCHEMBL4598959

CC(=O)NCCOc1cccc(CNc2c(Nc3ccc4nc[nH]c4c3)c(=O)c2=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 7/20 0.49
ROCK2 O75116 2/20 0.46
PLK4 O00444 1/20 0.46
CHEK1 O14757 1/20 0.46
DAPK3 O43293 1/20 0.46
DYRK3 O43781 1/20 0.46
JAK2 O60674 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
CHEK2 O96017 1/20 0.46
PRKCG P05129 1/20 0.46
CDK1 P06493 1/20 0.46
ROS1 P08922 1/20 0.46
PIM1 P11309 1/20 0.46
PRKACA P17612 1/20 0.46
RPS6KB1 P23443 1/20 0.46
CDK2 P24941 1/20 0.46
MAPK1 P28482 1/20 0.46
AKT1 P31749 1/20 0.46
AKT2 P31751 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4908299 0.93 ROCK2 (0.48) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4598622 0.86 QPCT (0.50) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4599132 0.85 QPCT (0.47) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4907508 0.82 QPCT (0.46) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4596911 0.81 NAMPT (0.47) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4598322 0.81 ROCK2 (0.44) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4905319 0.81 QPCT (0.46) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4597195 0.80 ROCK2 (0.44) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4599119 0.80 ROCK2 (0.41) QPCTROCK2PLK4CHEK1DAPK3
SCHEMBL4906532 0.78 ROCK2 (0.45) QPCTROCK2PLK4CHEK1DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed