SCHEMBL4598966

SCHEMBL4598966

O=c1c(NCc2cccc(O)c2F)c(Nc2ccc3nc[nH]c3c2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.42
CDC7 O00311 1/20 0.41
PLK4 O00444 1/20 0.41
CHEK1 O14757 1/20 0.41
DAPK3 O43293 1/20 0.41
RPS6KA5 O75582 1/20 0.41
MAP4K4 O95819 1/20 0.41
CHEK2 O96017 1/20 0.41
PIM1 P11309 1/20 0.41
PRKACA P17612 1/20 0.41
RPS6KB1 P23443 1/20 0.41
AKT1 P31749 1/20 0.41
AKT2 P31751 1/20 0.41
FLT4 P35916 1/20 0.41
PRKCI P41743 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
RPS6KA3 P51812 1/20 0.41
PRKCD Q05655 1/20 0.41
PRKAA1 Q13131 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4902107 0.92 ROCK1 (0.41) CDK1CDC7PLK4CHEK1DAPK3
SCHEMBL4596911 0.81 NAMPT (0.47) CDK1PLK4CHEK1DAPK3RPS6KA5
SCHEMBL4898762 0.81 ROCK1 (0.41) CDK1CDC7PLK4CHEK1DAPK3
SCHEMBL4898774 0.80 ROCK1 (0.43) CDK1CDC7PLK4CHEK1DAPK3
SCHEMBL4598446 0.80 ROCK1 (0.40) CDK1CDC7PLK4CHEK1DAPK3
SCHEMBL14066719 0.79 IP6K1 (0.55) CDK1PLK4CHEK1DAPK3MAP4K4
SCHEMBL4907489 0.76 ROCK1 (0.39) CDK1CDC7PLK4CHEK1DAPK3
SCHEMBL28651280 0.76 QPCT (0.57) QPCTNAMPTADRA2AADRA2CADRA1D
SCHEMBL4598825 0.76 QPCT (0.47) CDK1PLK4CHEK1DAPK3MAP4K4
SCHEMBL4905527 0.76 ROCK1 (0.42) CDK1CDC7PLK4CHEK1DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed