SCHEMBL4598825

SCHEMBL4598825

O=c1c(NCCc2cccc(O)c2)c(Nc2ccc3nc[nH]c3c2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 6/20 0.47
NAMPT P43490 1/20 0.46
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
ATM Q13315 1/20 0.43
ADRA2A P08913 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
MELK Q14680 1/20 0.41
EPHX1 P07099 1/20 0.39
F2 P00734 1/20 0.39
PRSS1 P07477 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
STAT6 P42226 1/20 0.38
P2RY14 Q15391 1/20 0.38
PAK4 O96013 1/20 0.38
KDR P35968 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4904991 0.92 ROCK2 (0.39) QPCTNAMPTTP53MAPTRAB9A
SCHEMBL4596911 0.89 NAMPT (0.47) QPCTNAMPTTP53MAPTRAB9A
SCHEMBL4905587 0.81 ROCK1 (0.48) QPCTNAMPTKDRPDGFRBIP6K1
SCHEMBL4597942 0.81 KDR (0.40) QPCTRAB9AF2PRSS1L3MBTL1
SCHEMBL14066719 0.80 IP6K1 (0.55) QPCTNAMPTTP53MAPTRAB9A
SCHEMBL4598401 0.79 KDR (0.47) QPCTNAMPTTP53MAPTRAB9A
SCHEMBL4597328 0.77 AURKB (0.47) QPCTNAMPTTP53MAPTRAB9A
SCHEMBL4373012 0.76 FLT4 (0.60) KDRPLK4CHEK1DAPK3ROCK2
SCHEMBL30673017 0.76 TBXA2R (0.47) KDRCHEK1MAP4K4CHEK2PRKCG
SCHEMBL4598966 0.76 CDK1 (0.42) QPCTNAMPTTP53MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed