SCHEMBL4599400

SCHEMBL4599400

Cc1ccc(NC(=O)/C=C/c2ccncc2)cc1C(=O)Nc1ccc2[nH]c(-c3ccccc3)nc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 4/20 0.51
MMP13 P45452 4/20 0.51
MAOB P27338 1/20 0.48
BTK Q06187 1/20 0.48
NR2E3 Q9Y5X4 1/20 0.47
MAPT P10636 5/20 0.46
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 4/20 0.46
HTT P42858 3/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
RAB9A P51151 5/20 0.44
POLB P06746 3/20 0.44
NPC1 O15118 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4614189 0.95 MAOB (0.54) MMP2MMP13MAOBBTKNR2E3
SCHEMBL4614145 0.91 BTK (0.50) MMP2MMP13MAOBBTKNR2E3
SCHEMBL1136425 0.89 BTK (0.52) MMP2MMP13MAOBBTKNR2E3
SCHEMBL1136426 0.89 BTK (0.52) MMP2MMP13MAOBBTKNR2E3
SCHEMBL13836664 0.84 MMP2 (0.61) MMP2MMP13MAOBMAPTKDM4E
SCHEMBL13836663 0.84 MMP2 (0.61) MMP2MMP13MAOBMAPTKDM4E
SCHEMBL8767799 0.84 MMP2 (0.61) MMP2MMP13MAOBMAPTKDM4E
SCHEMBL1136434 0.83 BTK (0.57) MMP2MMP13MAOBBTKNR2E3
SCHEMBL1136433 0.83 BTK (0.57) MMP2MMP13MAOBBTKNR2E3
SCHEMBL13836049 0.81 POLB (0.60) MMP2MMP13MAOBMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919910-A1 AZABENZIMIDAZOLE DERIVATIVES, THEIR MANUFACTURE AND USE AS ANTI-CANCER AGENTS F. Hoffmann-la Roche AG (CH) 2008-05-14 EP claimed
WO-2007017143-A1 AZABENZIMIDAZOLE DERIVATIVES, THEIR MANUFACTURE AND USE AS ANTI-CANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2007-02-15 WO claimed