SCHEMBL4600173

SCHEMBL4600173

CCN(CCN(c1ccc(OC)nc1)S(=O)(=O)c1ccccc1C(=O)O)C(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.51
HCRTR2 O43614 3/20 0.51
OXTR P30559 13/20 0.44
KMT2A Q03164 2/20 0.39
TAS2R14 Q9NYV8 1/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.38
AVPR1A P37288 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4459186 0.93 HCRTR1 (0.49) HCRTR1HCRTR2OXTRKMT2ATAS2R14
SCHEMBL4470460 0.90 HCRTR2 (0.62) HCRTR1HCRTR2OXTRAVPR1A
SCHEMBL4457211 0.88 HCRTR1 (0.50) HCRTR1HCRTR2OXTRLMNAAVPR1A
SCHEMBL4459456 0.86 HCRTR1 (0.49) HCRTR1HCRTR2OXTRTAS2R14LMNA
SCHEMBL4461806 0.84 HCRTR2 (0.61) HCRTR1HCRTR2OXTRAVPR1A
SCHEMBL4464707 0.84 KMT2A (0.52) HCRTR1HCRTR2OXTRKMT2ALMNA
SCHEMBL4457691 0.84 OXTR (0.56) HCRTR1HCRTR2OXTRKMT2ALMNA
SCHEMBL4453885 0.84 HCRTR2 (0.46) HCRTR1HCRTR2OXTRTAS2R14LMNA
SCHEMBL4455651 0.83 HCRTR2 (0.57) HCRTR1HCRTR2OXTRAVPR1A
SCHEMBL4457194 0.83 HCRTR2 (0.47) HCRTR1HCRTR2OXTRTAS2R14LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912655-A2 AMINOETHANE SULFONAMIDE OREXIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2008-04-23 EP claimed
WO-2007019234-A2 AMINOETHANE SULFONAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-02-15 WO claimed