SCHEMBL4600253

SCHEMBL4600253

CCOc1cc(C(F)(F)F)ccc1C(=O)NC1Cc2cc(OCC(F)(F)F)c(S(=O)(=O)Nc3cnc(C(C)C)s3)cc2C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
CSF1R P07333 1/20 0.35
CCR2 P41597 3/20 0.32
CRHR1 P34998 1/20 0.32
APOB P04114 1/20 0.32
MTTP P55157 1/20 0.32
PRMT5 O14744 1/20 0.32
IDH2 P48735 1/20 0.32
CNR2 P34972 1/20 0.32
SCN8A Q9UQD0 2/20 0.32
SCN10A Q9Y5Y9 2/20 0.32
KCNH2 Q12809 2/20 0.32
MCL1 Q07820 1/20 0.31
KDM5A P29375 1/20 0.31
ALPL P05186 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
USP2 O75604 1/20 0.31
CCRL2 O00421 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1967111 0.89 ALDH1A1 (0.41) ALDH1A1POLBCRHR1APOBMTTP
SCHEMBL1970540 0.82 ALDH1A1 (0.41) ALDH1A1USP2
SCHEMBL1971306 0.80 ALDH1A1 (0.42) ALDH1A1SCN8AUSP2
SCHEMBL1970268 0.80 ALDH1A1 (0.41) ALDH1A1CRHR1MCL1USP2
SCHEMBL1971486 0.77 ALDH1A1 (0.42) ALDH1A1POLBUSP2
SCHEMBL1969955 0.73 ALDH1A1 (0.40) ALDH1A1KCNH2MCL1USP2
SCHEMBL1969957 0.73 ALDH1A1 (0.40) ALDH1A1KCNH2MCL1USP2
SCHEMBL1973043 0.73 ALDH1A1 (0.40) ALDH1A1KCNH2MCL1USP2
SCHEMBL1970190 0.71 SCN9A (0.40) USP2
SCHEMBL1969717 0.70 ALDH1A1 (0.39) ALDH1A1POLBALPLUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937675-A2 BICYCLIC ARYL-SULFONIC ACID [1,3,4]-THIADIAZOL-2-YL-AMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS Sanofi-Aventis (FR) 2008-07-02 EP disclosed
WO-2007039174-A2 BICYCLIC ARYL-SULFONIC ACID [1,3,4]-THIADIAZOL-2-YL-AMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed