SCHEMBL4600817

SCHEMBL4600817

CC(=O)C(c1ccccc1)c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.54
SLC6A4 P31645 2/20 0.54
SLC6A3 Q01959 2/20 0.54
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 3/20 0.45
POLB P06746 2/20 0.45
MAPT P10636 1/20 0.45
KDM4E B2RXH2 2/20 0.44
HSD17B10 Q99714 1/20 0.44
TSHR P16473 1/20 0.44
ROCK2 O75116 1/20 0.44
RPS6KA5 O75582 1/20 0.44
MAP4K4 O95819 1/20 0.44
CDK1 P06493 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL396389 0.87 L3MBTL1 (0.56) TDP1L3MBTL1KMT2ALMNAALDH1A1
Benzene SCHEMBL27414119 0.87 L3MBTL1 (0.56) TDP1L3MBTL1KMT2ALMNAALDH1A1
Bicarbonate SCHEMBL28144656 0.85 L3MBTL1 (0.54) TDP1L3MBTL1KMT2ALMNAALDH1A1
SCHEMBL27924002 0.85 L3MBTL1 (0.54) TDP1L3MBTL1KMT2ALMNAALDH1A1
SCHEMBL29024912 0.85 L3MBTL1 (0.54) TDP1L3MBTL1KMT2ALMNAALDH1A1
SCHEMBL17710384 0.85 L3MBTL1 (0.54) TDP1L3MBTL1KMT2ALMNAALDH1A1
Bicarbonate SCHEMBL19031939 0.85 L3MBTL1 (0.54) TDP1L3MBTL1KMT2ALMNAALDH1A1
SCHEMBL6803687 0.83 SLC6A2 (0.58) SLC6A2SLC6A4SLC6A3TDP1L3MBTL1
SCHEMBL14284024 0.83 SMN1; SMN2 (0.55) SLC6A2SLC6A4SLC6A3HTTSMN1; SMN2
SCHEMBL28787356 0.83 MAPKAPK2 (0.46) SLC6A3LMNAALDH1A1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1915361-A1 ALKYLPYRIDYL QUINOLINES AS NK3 RECEPTOR MODULATORS AstraZeneca AB (SE) 2008-04-30 EP claimed
WO-2007018466-A1 ALKYLPYRIDYL QUINOLINES AS NK3 RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-02-15 WO claimed
CN-105917215-A METHOD FOR ANALYSING A SAMPLE COMPRISING AT LEAST A FIRST AND A SECOND SCALE INHIBITOR 凯米罗总公司 2016-08-31 CN disclosed
EP-1915361-A1 ALKYLPYRIDYL QUINOLINES AS NK3 RECEPTOR MODULATORS AstraZeneca AB (SE) 2008-04-30 EP disclosed
WO-2007018466-A1 ALKYLPYRIDYL QUINOLINES AS NK3 RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-02-15 WO disclosed