SCHEMBL4601908

SCHEMBL4601908

CCCOc1ccc(-c2cc(F)cc(C(=O)O)c2)cc1C(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 5/20 0.49
ICAM1 P05362 5/20 0.49
ITGAL P20701 5/20 0.49
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MAPT P10636 3/20 0.41
HPGD P15428 3/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC3 O15379 3/20 0.40
HDAC4 P56524 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC7 Q8WUI4 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC10 Q969S8 3/20 0.40
HDAC11 Q96DB2 3/20 0.40
HDAC8 Q9BY41 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC9 Q9UKV0 3/20 0.40
HDAC5 Q9UQL6 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14564875 0.94 ITGB2 (0.49) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL14557654 0.94 ITGB2 (0.49) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL14557744 0.94 ITGB2 (0.47) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL4603045 0.92 ITGB2 (0.40) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14564912 0.91 HDAC3 (0.46) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL4600803 0.91 HDAC3 (0.46) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL14557666 0.90 ITGB2 (0.43) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL14159167 0.90 MAPT (0.47) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL14557640 0.88 ITGB2 (0.43) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL14564810 0.88 ITGB2 (0.43) ITGB2ICAM1ITGALMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912970-A2 ACYLTRYPTOPHANOLS FOR FERTILITY CONTROL Bayer Schering Pharma Aktiengesellschaft (DE) 2008-04-23 EP claimed
WO-2007017289-A2 ACYLTRYPTOPHANOLS FOR FERTILITY CONTROL BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-02-15 WO claimed